Patent · US Active

Anti-fibrotic compounds

US11014873B2 · kind B2 · utility

1Cited by
26References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 31, 2018
Grant dateMay 25, 2021
Priority date
Expiry dateJan 31, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Provided herein are anti-fibrotic compounds, in particular those of Formula (I), that inhibit the TGF-beta signaling pathway. Also provided are pharmaceutical compositions comprising the anti-fibrotic compounds, and methods of treating diseases or conditions associated with fibrosis, inflammation, and benign or malignant neoplastic diseases in a subject by administering a compound or composition described herein. (Formula (I))

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.