Patent · US Active

Application of methyl 4-[9-(6-aminopuryl)]-2(s)-hydroxybutyrate in preparation of medicament for treating psoriasis and vitiligo

US11045475B2 · kind B2 · utility

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Key dates

Filing dateJun 29, 2017
Grant dateJun 29, 2021
Priority date
Expiry dateAug 9, 2037

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/42
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Provided in the present invention is a use of methyl 4-[9-(6-aminopuryl)]-2(s)-hydroxybutyrate in the preparation of a medicament for treating psoriasis and vitiligo. More specifically, the present invention uses mice whose psoriasis is induced by an imiquimod cream to observe a changing condition in skin lesions on the psoriasis-like mice, according to a psoriasis skin lesion area of the mice and grading standards for disease severity; the present invention also observes a proportion of lymphocytes in the spleens and cytokines in skin lesion tissues of the mice. A good therapeutic effect may be obtained by treating typical cases of vitiligo with an ointment of methyl 4-[9-(6-aminopuryl)]-2(s)-hydroxybutyrate. Results show that methyl 4-[9-(6-aminopuryl)]-2(s)-hydroxybutyrate used in the present invention has a good therapeutic effect on psoriasis and vitiligo, as well as a favorable prospect in clinical application.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.