Patent · US Active

Pyrazole compounds and uses thereof

US11072599B2 · kind B2 · utility

1Cited by
1References
25Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 30, 2018
Grant dateJul 27, 2021
Priority date
Expiry dateJan 30, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides pyrazole derivatives of Formula (I), and in particular N1-(4-(5-(cyclopropylmethyl)-1-methyl-1H-pyrazol-4-yl) pyridin-2-yl)cyclohexane-1,4-diamine derivatives and related compounds as casein kinase 1 (CK1) and/or interleukin 1 receptor associated kinase 1 (IRAKI) inhibitors for treating cancer, inflammatory and immune related disorders.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.