Patent · US Active

Phthalazine derivatives as inhibitors of PARP1, PARP2, and/or tubulin useful for the treatment of cancer

US11072600B2 · kind B2 · utility

1Cited by
3References
42Claims
0Family size

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Key dates

Filing dateJun 23, 2017
Grant dateJul 27, 2021
Priority date
Expiry dateJun 23, 2037

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The application relates to phthalazine derivatives of formula (I) which are inhibitors of PARP1, PARP2 and/or tubulin and thus useful for the treatment of cancer. Also disclosed are pharmaceutical formulations containing such compounds, as well as combinations of these compounds with at least one additional therapeutic agent.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.