Patent · US Active

Solution phase synthesis and crystallization of beta-turn peptidomimetic cyclic salts

US11078234B2 · kind B2 · utility

2Cited by
1References
21Claims
0Family size

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Key dates

Filing dateNov 8, 2018
Grant dateAug 3, 2021
Priority date
Expiry dateNov 8, 2038

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

The present disclosure relates to methods of preparing and crystallizing β-turn cyclic peptidomimetic salts of formula I: where R1, R2, R3, R4, R5, R6, R7, R8, R10, X, Y and n are as defined in the specification. The present disclosure provides a more efficient route for preparing a crystalline form of β-turn cyclic peptidomimetic compounds and salts thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.