Patent · US Active

Catalyst-free and redox-neutral innate trifluoromethylation and alkylation of (hetero)aromatics enabled by light

US11098036B2 · kind B2 · utility

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12Claims
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Assignee

Inventors

Key dates

Filing dateSep 28, 2018
Grant dateAug 24, 2021
Priority date
Expiry dateSep 28, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2602/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present disclosure relates to reagents and method for performing trifluoromethylation, difluoromethylation or alkylation of aromatic or heteroaromatic rings in a redox-neutral manner without any catalyst which are enabled by light. In addition, there are methods for synthesizing the starting reagents used in the trifluoromethylation, difluoromethylation or alkylation reactions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.