Patent · US Active

Bisphenol derivatives and their use as androgen receptor activity modulators

US11142508B2 · kind B2 · utility

4Cited by
29References
24Claims
0Family size

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Key dates

Filing dateApr 14, 2020
Grant dateOct 12, 2021
Priority date
Expiry dateApr 14, 2040

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D233/60
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having a structure of Formula I or a pharmaceutically acceptable salt, tautomer or stereoisomer thereof, wherein R1, R2, R3, R11a, R11b, R11c, R11d, and X, are as defined herein, are provided. Uses of such compounds for modulating androgen receptor activity, imaging diagnostics in cancer and therapeutics, and methods for treatment of subjects in need thereof, including prostate cancer are also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.