Patent · US Active

3,3-difluoroallylamines or salts thereof and pharmaceutical compositions comprising the same

US11168073B2 · kind B2 · utility

3Cited by
2References
32Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 12, 2019
Grant dateNov 9, 2021
Priority date
Expiry dateDec 12, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D498/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present technology provides 3,3-difluoroallylamines or pharmaceutically acceptable salts thereof, preparation processes thereof, pharmaceutical compositions comprising the same, and uses thereof. The 3,3-difluoroallylamines or their pharmaceutically acceptable salts exhibit potent inhibitory activity on VAP-1 and therefore can be usefully applied, e.g., for the treatment and prophylaxis of nonalcoholic hepatosteatosis (NASH).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.