Patent · US Active

Small molecule inhibitors of NF-κB inducing kinase

US11254673B2 · kind B2 · utility

1Cited by
3References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 29, 2020
Grant dateFeb 22, 2022
Priority date
Expiry dateAug 18, 2040

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to compounds that inhibit NIK and pharmaceutical compositions comprising such compounds and methods of using the same. These compounds and pharmaceutical compositions are envisaged to be useful for preventing or treating diseases such as cancer (such as B-cell malignancies including leukemias, lymphomas and myeloma), inflammatory disorders, autoimmune disorders, immunodermatologic disorders such as palmoplantar pustulosis and hidradenitis suppurativa, and metabolic disorders such as obesity and diabetes.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.