Patent · US Active

Synthesis of key intermediate of KRAS G12C inhibitor compound

US11299491B2 · kind B2 · utility

12Cited by
50References
1Claims
0Family size

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Key dates

Filing dateNov 15, 2019
Grant dateApr 12, 2022
Priority date
Expiry dateFeb 1, 2040

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C309/24
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to an improved, efficient, scalable process to prepare intermediate compounds, such as compound 5M, having the structure useful for the synthesis of compounds that target KRAS G12C mutations, such as

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.