Patent · US Active

Stable amorphous form of sacubitril valsartan trisodium complex and processes for preparation thereof

US11318116B2 · kind B2 · utility

0Cited by
2References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 22, 2020
Grant dateMay 3, 2022
Priority date
Expiry dateSep 22, 2040

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to stable amorphous form of sacubitril valsartan trisodium complex and its solid dispersion compounds, processes for their preparation and pharmaceutical composition comprising the same. The present invention also relates to an improved process for the preparation of sacubitril sodium and its use in the preparation of sacubitril valsartan trisodium complex.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.