Patent · US Active

Crystalline forms of Acalabrutinib

US11345706B2 · kind B2 · utility

0Cited by
1References
9Claims
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Assignee

Inventors

Key dates

Filing dateAug 23, 2018
Grant dateMay 31, 2022
Priority date
Expiry dateSep 6, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides crystalline forms of Acalabrutinib, Specific crystalline forms provided by the present invention include Acalabrutinib Form APO-I, a co-crystal of Acalabrutinib and urea; APO-II, a co-crystal of Acalabrutinib and nicotinamide; APO-III, a co-crystal of Acalabrutinib and L-sorbitol; APO-IV, a crystalline form of Acalabrutinib; and APO-V, a co-crystal of Acalabrutinib and urea.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.