Patent · US Active

Tryptophan hydroxylase inhibitor and pharmaceutical composition including same

US11407763B2 · kind B2 · utility

0Cited by
0References
20Claims
0Family size

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Inventors

Key dates

Filing dateAug 24, 2018
Grant dateAug 9, 2022
Priority date
Expiry dateAug 29, 2038

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a novel tryptophan hydroxylase inhibitor and a pharmaceutical composition including same, wherein the novel tryptophan hydroxylase inhibitor has an excellent inhibitory effect on TPH1, and thus can be usefully used for the prevention or treatment of disorders, such as metabolic disorders, cancer, digestive or cardiovascular system disorders, related to TPH1 activity. In particular, the novel tryptophan hydroxylase inhibitor has an excellent treatment effect on inflammatory bowel disorders, and thus can be usefully used for the treatment of inflammatory bowel disorder.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.