Patent · US Active

Inhibitors of KEAP1-Nrf2 protein-protein interaction

US11427601B1 · kind B1 · utility

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4References
44Claims
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Key dates

Filing dateAug 30, 2021
Grant dateAug 30, 2022
Priority date
Expiry dateAug 30, 2041

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Sultam compounds, pharmaceutical compositions containing them, methods of making them, and methods of using them including methods for treating disease states, disorders, and conditions associated with the KEAP1-Nrf2 interaction, such as inflammatory bowel disease, including Crohn's disease and ulcerative colitis.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.