Patent · US Active

Process for preparing soluble guanylate cyclase stimulators

US11466014B2 · kind B2 · utility

1Cited by
0References
11Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMar 7, 2019
Grant dateOct 11, 2022
Priority date
Expiry dateMar 17, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention relates to novel methods for preparing 3-substituted 1,2,4-triazole compounds of Formula IA: as sGC stimulators. The method comprises reacting the amidrazone compound represented by Formula IIA: or a salt thereof, with a carboxylic acid, an activated ester, a thioester, an acid halide, a thioacyl halide, or an acid anhydride in the presence of a base.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.