Patent · US Active

Substituted 1,2-oxaborolan-2-ols as PDE4 inhibitors

US11559538B2 · kind B2 · utility

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Assignee

Inventors

Key dates

Filing dateOct 28, 2020
Grant dateJan 24, 2023
Priority date
Expiry dateJul 21, 2041

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to boron containing compounds of Formula (IA): that inhibit phosphodiesterase 4 (PDE4). The invention also encompasses pharmaceutical compositions containing these compounds and methods for treating diseases, conditions, or disorders ameliorated by inhibition of PDE4.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.