Polymorphs of ARRY-380, a selective HER2 inhibitor and pharmaceutical compositions containing them
US11571424B2 · kind B2 · utility
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19Claims
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Key dates
| Filing date | Jul 29, 2020 |
| Grant date | Feb 7, 2023 |
| Priority date | — |
| Expiry date | Jul 29, 2040 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D471/04
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Polymorphs of N4-(4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)-3-methylphenyl)-N6-(4,4-dimethyl-4,5-dihydrooxazol-2-yl)quinazoline-4,6-diamine are provided herein. Processes for preparing the polymorphs and pharmaceutical composition comprising the polymorphs are also disclosed.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.