Patent · US Active

Synthetic method for the preparation of a 3-[5-amino-4-(3-cyanobenzoyl)-pyrazol compound

US11649213B2 · kind B2 · utility

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2References
17Claims
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Assignee

Inventors

Key dates

Filing dateSep 26, 2019
Grant dateMay 16, 2023
Priority date
Expiry dateDec 19, 2039

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D231/38
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Provided is a process for preparing a compound, comprising the steps of a) Reacting a compound of Formula A (Formula A) with the compound 3 (3) to provide the compound 5 (5) or a salt or solvate thereof, wherein R is a linear or branched C1-C5 alkyl. Further provided is the compound 5 or a salt or solvate thereof. (5) The use of these compounds in the synthesis of 3-[5-Amino-4-(3-Cyanobenzoyl)-Pyrazol-1-yl]-N-Cyclopropyl-4-Methylbenzamide is also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.