Patent · US Active

Pharmaceutical composition containing quinoline derivative

US11701349B2 · kind B2 · utility

0Cited by
3References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 23, 2018
Grant dateJul 18, 2023
Priority date
Expiry dateJun 26, 2039

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/1694
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides a pharmaceutical composition comprising (R, E)-N-(4-(3-chloro-4-(pyridin-2-ylmethoxy) phenylamino)-3-cyano-7-ethoxyquinolin-6-yl)-3-(1-methylpyrrolidinyl-2-yl)-acrylamide or a pharmacologically acceptable salt thereof, which is obtained by mixing the quinoline derivative or a pharmacologically acceptable salt thereof, a wetting agent, a disintegrant, and at least one pharmaceutical excipient; granulating; dynamic drying; and optionally compressing into tablets or filling into capsules after mixing with a lubricant.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.