Patent · US Active

Polymorphs of sepiapterin and salts thereof

US11773097B2 · kind B2 · utility

5Cited by
25References
17Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJun 9, 2021
Grant dateOct 3, 2023
Priority date
Expiry dateDec 4, 2041

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed are crystalline forms of sepiapterin free base selected from polymorphs A, B, C, D, E, F, and G, and combinations thereof, as well as crystalline polymorphs of salts of sepiapterin. Also disclosed are pharmaceutical compositions containing one or more such polymorphs and methods for preparing such polymorphs. Sepiapterin is useful in the treatment of a number diseases associated with low cellular levels of BH4, for example, phenylketonuria.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.