Substituted pyrrolidones and piperidones as small molecule inhibitors of EZH2 and EED protein binding
US11919855B2 · kind B2 · utility
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19Claims
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Key dates
| Filing date | Apr 29, 2022 |
| Grant date | Mar 5, 2024 |
| Priority date | — |
| Expiry date | Apr 29, 2042 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D207/27
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Disclosed are substituted pyrrolidones and piperidones which may be utilized as EZH2 targeting agents. The substituted pyrrolidones and piperidones may include substituted 2-pyrrolidones and 2-piperidones. The disclosed pyrrolidones and piperidones may be used in pharmaceutical compositions and methods for treating cell proliferative disorders such as cancer.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.