Patent · US Active

Rapafucin derivative compounds and methods of use thereof

US11945827B2 · kind B2 · utility

0Cited by
14References
4Claims
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Assignee

Inventors

Key dates

Filing dateMay 27, 2021
Grant dateApr 2, 2024
Priority date
Expiry dateAug 31, 2041

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/6561
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present disclosure provides macrocyclic compounds inspired by the immunophilin ligand family of natural products FK506 and rapamycin. The generation of a Rapafucin library of macrocyles that contain FK506 and rapamycin binding domains should have great potential as new leads for developing drugs to be used for treating diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.