Patent · US Active

Bicyclic 1,4-diazepanones and therapeutic uses thereof

US11981644B2 · kind B2 · utility

0Cited by
25References
27Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 5, 2021
Grant dateMay 14, 2024
Priority date
Expiry dateDec 29, 2041

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Provided herein are compounds of formula (1): or a stereoisomer or tautomer thereof, or a pharmaceutically acceptable salt of any of the foregoing, wherein X1, X2, Ry, Rz, R1, R2, R3, and R4 are as defined herein. Also provided herein is a pharmaceutically acceptable composition comprising a compound of formula (I), or a stereoisomer or tautomer thereof, or a pharmaceutically acceptable salt of any of the foregoing. Also provided herein are methods of using a compound of formula (I), or a stereoisomer or tautomer thereof, or a pharmaceutically acceptable salt of any of the foregoing, to treat various diseases, disorders, and conditions responsive to the modulation of the contractility of the skeletal sarcomere.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.