Patent · US Active

Bicyclic heterocyclyl derivatives as IRAK4 inhibitors

US11981685B2 · kind B2 · utility

1Cited by
11References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 28, 2023
Grant dateMay 14, 2024
Priority date
Expiry dateApr 28, 2043

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides bicyclic heterocyclyl kinase enzyme inhibitor compounds of formula (I), which are therapeutically useful as kinase inhibitors, particularly IRAK4 inhibitors. wherein A, Y, Z, X1, X2, X3, R1, R3, ‘m’, ‘n’ and ‘p’ have the meanings given in the specification and pharmaceutically acceptable salts or stereoisomers thereof that are useful in the treatment and prevention of diseases or disorders, in particular their use in diseases or disorders mediated by kinase enzyme, particularly IRAK4 enzyme. The present invention also provides pharmaceutical compositions comprising at least one of the compounds of compound of formula (I) together with a pharmaceutically acceptable carrier, diluent or excipient therefor.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.