Patent · US Active

Ligand regulated protein-protein interaction system

US12102653B2 · kind B2 · utility

0Cited by
3References
20Claims
0Family size

Assignees

Inventors

Key dates

Filing dateMay 4, 2023
Grant dateOct 1, 2024
Priority date
Expiry dateMay 4, 2043

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K2319/70
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A ligand regulated protein-protein interaction system based on a lipocalin-fold molecule including: (a) a lipocalin-fold molecule; (b) a lipocalin-fold ligand with a low molecular weight of 1500 Da or below; and (c) a lipocalin-fold binding interaction partner, wherein the lipocalin-fold molecule can bind to the lipocalin-fold ligand; and wherein the lipocalin-fold molecule bound to the lipocalin-fold ligand binds to the lipocalin-fold binding interaction partner with an affinity which is at least 10-fold higher than the affinity of the lipocalin-fold molecule not bound to the lipocalin-fold ligand; and wherein the lipocalin-fold binding interaction partner is not a naturally occurring protein which has an affinity of <10 μM to any naturally occurring lipocalin-fold molecule in the presence of any lipocalin-fold ligand.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.