Glutarimide-containing pan-KRAS-mutant degrader compounds and uses thereof
US12110291B2 · kind B2 · utility
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32Claims
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Key dates
| Filing date | Nov 30, 2023 |
| Grant date | Oct 8, 2024 |
| Priority date | — |
| Expiry date | Dec 1, 2043 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D519/00
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present disclosure relates to novel pan-KRAS glutarimide-containing compounds with KRAS degradation activities, pharmaceutical compositions containing such compounds, and their use in prevention and treatment diseases and conditions.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.