Patent · US Active

Crystal form a of NHE3 inhibitor, preparation method therefor and application thereof

US12122762B2 · kind B2 · utility

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20Claims
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Key dates

Filing dateSep 13, 2021
Grant dateOct 22, 2024
Priority date
Expiry dateJul 31, 2043

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Provided is crystal form A of N,N′-(10,17-dioxo-3,6,21,24-tetraoxa-9,11,16, 18-tetrazohexahexane-1,26-di-yl)bis(4-(6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinoline-4-yl) benzene sulfonamide. The crystal form has good light stability, high-temperature stability, and high-humidity stability.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.