Crystal form a of NHE3 inhibitor, preparation method therefor and application thereof
US12122762B2 · kind B2 · utility
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Key dates
| Filing date | Sep 13, 2021 |
| Grant date | Oct 22, 2024 |
| Priority date | — |
| Expiry date | Jul 31, 2043 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07B2200/13
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Provided is crystal form A of N,N′-(10,17-dioxo-3,6,21,24-tetraoxa-9,11,16, 18-tetrazohexahexane-1,26-di-yl)bis(4-(6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinoline-4-yl) benzene sulfonamide. The crystal form has good light stability, high-temperature stability, and high-humidity stability.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.