Patent · US Active

Compounds, compositions, and therapeutic uses thereof

US12145945B2 · kind B2 · utility

0Cited by
0References
4Claims
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Assignee

Inventors

Key dates

Filing dateMar 8, 2024
Grant dateNov 19, 2024
Priority date
Expiry dateMar 8, 2044

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to a compound of the Formula: and pharmaceutically salts thereof. The compound of the present invention inhibits Polθ. This novel therapeutic compound is therefore useful for the treatment and/or prevention of diseases and conditions in which Polθ activity is implicated, such as, for example but not limited to, the treatment and/or prevention of cancer. The present invention also relates to pharmaceutical compositions comprising the novel therapeutic compound defined herein, to processes for synthesising the compound and to their use for the treatment of diseases and/or conditions in which Polθ activity is implicated.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.