Patent · US Active

Crystalline and amorphous forms of a compound for the targeted degradation of estrogen receptor

US12162859B2 · kind B2 · utility

0Cited by
28References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 13, 2021
Grant dateDec 10, 2024
Priority date
Expiry dateSep 13, 2041

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present disclosure relates to polymorphic forms of (S)-3-(5-(4-((1-(4-((1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl)piperidin-4-yl)methyl)piperazin-1-yl)-1- oxoisoindolin-2-yl)piperidine-2,6-dione, methods of making these polymorphic forms, and compositions comprising these polymorphic forms. These polymorphic forms are useful in the treatment of various diseases, including, for example, breast cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.