Patent · US Active

Prostaglandin receptor EP2 antagonists, derivatives, and uses related thereto

US12240829B2 · kind B2 · utility

0Cited by
6References
2Claims
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Assignee

Inventors

Key dates

Filing dateMar 19, 2020
Grant dateMar 4, 2025
Priority date
Expiry dateMay 17, 2042

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The disclosure relates to Prostnglandin receptor EP2 antagonists, derivatives, compositions, and methods related thereto. In certain embodiments, the disclosure relates to methods of treating or preventing conditions and diseases in which EP2 receptor activation has a physiological role, such as but not limited to, brain injury, inflammatory diseases, epilepsy, neuroinflammation after a seizure, pain, endometriosis, cancer, rheumatoid arthritis, skin inflammation, vascular inflammation, colitis, and neurological disorders by administering a pharmaceutical composition comprising a compound disclosed herein to a subject in need thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.