Patent · US Active

Use of FAK inhibitor in preparation of drug for treating tumors having NRAS mutation

US12257251B2 · kind B2 · utility

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15Claims
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Assignee

Inventors

Key dates

Filing dateJul 11, 2023
Grant dateMar 25, 2025
Priority date
Expiry dateJul 11, 2043

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A use of a FAK inhibitor in the preparation of a drug for preventing and/or treating tumors having an NRAS mutation. A method for treating tumors that have experienced an NRAS mutation, which comprises administering an effective dose of a FAK inhibitor to an individual. A FAK inhibitor for treating tumors having an NRAS mutation. The FAK inhibitor is B1853520, defactinib, GSK2256098, PF-00562271, VS-4718 or a pharmaceutically acceptable salt thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.