Patent · US Active

Compositions and methods for treating EZH2-mediated cancer

US12274697B2 · kind B2 · utility

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6References
12Claims
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Key dates

Filing dateNov 1, 2022
Grant dateApr 15, 2025
Priority date
Expiry dateNov 1, 2042

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Methods for designing bivalent compounds which selectively degrade/disrupt EZH2 and compositions and methods of using such degraders/disruptors to treat EZH2-mediated cancer are provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.