Patent · US Active

Substituted 1-amino-1H-imidazole-5-carboxamide as Bruton's tyrosine kinase inhibitors

US12291516B2 · kind B2 · utility

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Inventors

Key dates

Filing dateMay 9, 2020
Grant dateMay 6, 2025
Priority date
Expiry dateJul 21, 2042

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/08
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed is a compound of formula I or a pharmaceutically acceptable salt, active metabolite, tautomer, stereoisomer, or prodrug thereof as BTK (Bruton's Tyrosine Kinase) inhibitors, which is useful for the treatment of autoimmune disease, inflammatory disease, cancer and potentially allergies.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.