Patent · US Active

Method of inhibiting TREM-1

US12370193B2 · kind B2 · utility

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1References
8Claims
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Key dates

Filing dateOct 1, 2021
Grant dateJul 29, 2025
Priority date
Expiry dateDec 22, 2043

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P29/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed herein are methods and uses of the polypharmacological modulator SR1903 and related compounds for inhibiting triggering receptor expressed on myeloid cells-1 (TREM-1) and treating diseases and conditions that are related to or mediated by TREM-1, such as inflammatory diseases, autoimmune diseases, metabolic disorders, and castration resistant prostate cancer (CRPC).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.