Patent · US Active

Phenylalanine-based LAT1 inhibitors and uses thereof

US12427124B1 · kind B1 · utility

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7References
28Claims
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Key dates

Filing dateFeb 25, 2025
Grant dateSep 30, 2025
Priority date
Expiry dateFeb 25, 2045

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2602/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Phenylalanine-based inhibitors of the Large Amino Acid Transporter 1 (LAT1) are disclosed. The compounds are useful in modulating the transcellular transport of substrates of LAT1 such as large neutral amino acids. The compounds are useful in immunomodulation therapies.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.