Patent · US Active

2,4-disubstituted pyrimidine derivative, preparation method therefor and use thereof

US12428394B2 · kind B2 · utility

0Cited by
3References
27Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJun 28, 2020
Grant dateSep 30, 2025
Priority date
Expiry dateJan 30, 2043

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention belongs to the field of chemical medicines, and particularly relates to a 2,4-disubstituted pyrimidine derivative, a preparation method therefor and a use thereof. The present invention provides a 2,4-disubstituted pyrimidine derivative, the structural formula of which is as shown in formula I. The present invention also provides a preparation method for the 2,4-disubstituted pyrimidine derivative and a use thereof. The 2,4-disubstituted pyrimidine derivative provided by the present invention can be used as a kinase inhibitor with double functional targets of JAK2 and FLT3, or a kinase inhibitor with independent functional targets of JAK2 or FLT3, thus providing a new choice for preparing a multi-target inhibitor.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.