Patent · US Active

Acetylation writer inhibitor development and uses thereof

US12428412B2 · kind B2 · utility

0Cited by
0References
30Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 1, 2019
Grant dateSep 30, 2025
Priority date
Expiry dateApr 29, 2042

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12N15/09
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed are bifunctional compounds (degraders) that target HAT EP300 for degradation. Also disclosed are pharmaceutical compositions containing the degraders and methods of using the compounds to treat disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.