Patent · US Expired

Vincamine derivatives and process for the preparation of vincamine and derivatives thereof

US3937709A · kind A · utility

10Cited by
3References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 15, 1973
Grant dateFeb 10, 1976
Priority date
Expiry dateJun 15, 1993

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D461/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

New compounds having the formula ##SPC1## In which Y represents a hydrogen atom, in which case Z.sub.1 and Z.sub.2 represent simultaneously an oxygen atom, or Z.sub.1 represents a methoxycarbonyl radical and Z.sub.2 a hydroxy radical, or Y and Z.sub.2 form together a carbon-carbon bond and Z.sub.1 is a methoxycarbonyl radical, said compounds being additionally characterized by a cis-fusion of the D/E rings. Said new compounds and vincamine and certain of its derivatives are prepared from an enamine having the formula: ##SPC2## In which R is H or C.sub.2 H.sub.5.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.