Patent · US Expired

Process for preparing cephalosporin compounds from 7-ADCA

US3957773A · kind A · utility

6Cited by
5References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 2, 1974
Grant dateMay 18, 1976
Priority date
Expiry dateJul 2, 1994

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D501/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

7.beta.-Amino-3-methylceph-3-em-4-carboxylic acid is converted to cephalexin in high yield and relatively uncontaminated with unreacted 7.beta.-amino-3-methylceph-3-em-4-carboxylic acid if it is silylated prior to acylation with phenyl glycyl chloride hydrochloride and if the acylation reaction is conducted in dimethylformamide at low temperature in the presence of certain weak tertiary nitrogen bases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.