Patent · US Expired

Substituted nitrobenzophenone derivatives

US3957777A · kind A · utility

4Cited by
0References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 3, 1974
Grant dateMay 18, 1976
Priority date
Expiry dateJul 3, 1994

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

New compounds of the formula (I), ##SPC1## wherein PA1 R.sub.1 and R.sub.2 each stand for a saturated or unsaturated, straightchained or branched alkyl group, an aralkyl group, a saturated or unsaturated cycloalkyl group or an aryl group, or PA1 R.sub.1 and R.sub.2 together with the adjacent nitrogen atom form a substituted or unsubstituted heterocyclic group which can contain a further oxygen or nitrogen hetero atom, But when R.sub.1 is methyl, R.sub.2 is a group other than methyl, are prepared by reacting a compound of the formula (II), ##SPC2## wherein X stands for halogen, with a secondary amine of the general formula (III), EQU r.sub.1 --nh--r.sub.2. (iii) the new compounds of the general formula (I), as well as their pharmaceutical acceptable acid addition salts or quaternary ammonium salts are active primarily in the induction of liver microsomal enzyme, but they also possess antipyretic activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.