Patent · US Expired

N-(1-(1,3-D ihydro-1,3-dioxo-2H-benz(de)-isoquinolin-2-yl)alkyl)-4-N-piperidinyl)-n-p henylalkylamides

US3959286A · kind A · utility

10Cited by
2References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 6, 1975
Grant dateMay 25, 1976
Priority date
Expiry dateJan 6, 1995

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the following formula and their acid addition salts ##SPC1## Wherein R.sup.1 and R.sup.2 are independently selected from hydrogen, halogen, lower alkyl, lower alkoxy, lower alkylthio, nitro, cyano, amino and trifluoromethyl; A is a straight or branched chain alkylene of 1 to 8 carbons; R.sup.3 is phenyl or substituted phenyl; and R is lower alkyl or cycloalkyl of 3 to 7 carbons are disclosed. These compounds exhibit antidepressant activity. In addition these compounds are useful as antiinflammatory agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.