N-(1-(1,3-D ihydro-1,3-dioxo-2H-benz(de)-isoquinolin-2-yl)alkyl)-4-N-piperidinyl)-n-p henylalkylamides
US3959286A · kind A · utility
Assignee
Inventors
Key dates
| Filing date | Jan 6, 1975 |
| Grant date | May 25, 1976 |
| Priority date | — |
| Expiry date | Jan 6, 1995 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D401/06
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Compounds of the following formula and their acid addition salts ##SPC1## Wherein R.sup.1 and R.sup.2 are independently selected from hydrogen, halogen, lower alkyl, lower alkoxy, lower alkylthio, nitro, cyano, amino and trifluoromethyl; A is a straight or branched chain alkylene of 1 to 8 carbons; R.sup.3 is phenyl or substituted phenyl; and R is lower alkyl or cycloalkyl of 3 to 7 carbons are disclosed. These compounds exhibit antidepressant activity. In addition these compounds are useful as antiinflammatory agents.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.