Oxazinoindole- and thiazinoindole derivatives
US3962236A · kind A · utility
Assignee
Inventors
Key dates
| Filing date | May 28, 1974 |
| Grant date | Jun 8, 1976 |
| Priority date | — |
| Expiry date | May 28, 1994 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D209/08
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Oxazinoindole derivatives characterized by having an amino(lower)alkyl radical attached to the 1 position of a 1H-1,4-oxazino[4,3-a]indole nucleus are disclosed. The amino portion of the amino(lower)alkyl radical may be further substituted with one or two lower alkyl groups or incorporated in a heterocyclic amine radical. The derivatives are substituted further at positions 1 and 10 and may be optionally substituted at positions 3, 4, 6, 7, 8 and 9. The oxazinoindole derivatives of this invention are useful antidepressant and antiulcer agents. Methods for the preparation and use of these derivatives are also disclosed.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.