Patent · US Expired

Oxazinoindole- and thiazinoindole derivatives

US3962236A · kind A · utility

1Cited by
3References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 28, 1974
Grant dateJun 8, 1976
Priority date
Expiry dateMay 28, 1994

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D209/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Oxazinoindole derivatives characterized by having an amino(lower)alkyl radical attached to the 1 position of a 1H-1,4-oxazino[4,3-a]indole nucleus are disclosed. The amino portion of the amino(lower)alkyl radical may be further substituted with one or two lower alkyl groups or incorporated in a heterocyclic amine radical. The derivatives are substituted further at positions 1 and 10 and may be optionally substituted at positions 3, 4, 6, 7, 8 and 9. The oxazinoindole derivatives of this invention are useful antidepressant and antiulcer agents. Methods for the preparation and use of these derivatives are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.