Patent · US Expired

Method for making a microsealed delivery device

US3992518A · kind A · utility

139Cited by
8References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 29, 1975
Grant dateNov 16, 1976
Priority date
Expiry dateSep 29, 1995

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/2036
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention is concerned with a pharmaceutical delivery device comprising a biologically acceptable silicone polymer matrix having microsealed compartments of 10-200 microns throughout, wherein the microsealed compartments contain a pharmaceutical in a hydrophilic solvent system. The biologically acceptable silicone polymer matrix is formed by in situ cross linking of a liquid, biologically acceptable silicone polymer in an emulsion of pharmaceutical in the hydrophilic solvent system and liquid biologically acceptable silicone polymer. The biologically acceptable silicone polymer matrix is placed in a sealed or unsealed biologically acceptable polymer container. The rate of release of pharmaceutical is controlled by altering the solubility characteristics of the hydrophilic solvent system and/or the biologically acceptable polymer matrix, the rate of release being independent of time when the ratio of the partition coefficient of the pharmaceutical between the hydrophilic solvent system and biologically acceptable silicone polymer matrix to the solubility of the pharmaceutical in the hydrophilic solvent system is between 1 and 10.sup.-.sup.4 ml/mcg.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.