Imidazolylacetic acid amides

US3993647A · kind A · utility

Assignee

• BAYER HEALTHCARE LLC · DE

Inventors

• Jurgen Wenzelburger
• Karl H. Buchel · Burscheid, DE
• Manfred Plempel · Haan, DE
• Werner Meiser

Key dates

• Filing date: Jul 9, 1975
• Grant date: Nov 23, 1976
• Expiry date: Jul 9, 1995

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D417/06
• WIPO field: Pharmaceuticals
• WIPO sector: Chemistry

Abstract

Imidazolylacetic acid amides of the formula: ##SPC1## Or pharmaceutically acceptable nontoxic salts thereof wherein Either R.sup.1 is phenyl or cycloalkyl, unsubstituted or substituted by one or more substituents; and R.sup.2 is hydrogen; Or R.sup.1 and R.sup.2, together with the nitrogen atom to which they are attached, form a saturated 5 to 7-membered heterocyclic ring which ring may contain an --SO.sub.2 -- or --NY-- moiety wherein Y is alkoxycarbonyl, dialkylaminocarbonyl, or phenyl or diphenylmethyl, unsubstituted or substituted by one or more substituents and wherein said 5 to 7-membered heterocyclic ring itself is otherwise unsubstituted or substituted by one or more substituents; and X.sup.1, x.sup.2, x.sup.3 and X.sup.4 are the same or different and are each hydrogen or halogen, Are antimycotic agents.