Patent · US Expired

Xanthone-2-carboxylic acid compounds

US4024276A · kind A · utility

1Cited by
1References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 1, 1975
Grant dateMay 17, 1977
Priority date
Expiry dateJul 1, 1995

Classification

  • Technology area (CPC G)Physics
  • CPC primaryG21F1/125
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel xanthone-2-carboxylic acid compounds of the formula ##STR1## wherein A is selected from the group consisting of --COOR', a 1H-tetrazol-5-yl and a 1H-tetrazolylcarbamoyl, R' is selected from the group consisting of hydrogen, alkyl of 1 to 5 carbon atoms and cation of a non-toxic, pharmaceutically acceptable organic or inorganic base, R is selected from the group consisting of hydrogen, alkyl of 1 to 9 carbon atoms, alkoxy of 1 to 9 carbon atoms and alkoxy alkoxy of 2 to 9 carbon atoms and X is selected from the group consisting of ##STR2## AND ##STR3## WHEREIN R.sub.1 is alkyl of 1 to 5 carbon atoms, R.sub.2 is selected from the group consisting of hydrogen, acyl of an aliphatic acid of 1 to 5 carbon atoms, aroyl of 7 to 8 carbon atoms, araliphatic acyl with 1 to 5 carbon atoms in the aliphatic portion and 6 or 7 carbon atoms in the aryl portion, aralkyl of 7 to 8 carbon atoms, arylsulfonyl, a carbamoyl, a carboxyalkyl of 1 to 5 carbon atoms, --CO--(CH.sub.2).sub.n -- Het where n is 1, 2 or 3 and Het is a N-attached nitrogen heterocyclic which may contain an additional heteroatom and ##STR4## AND Alk is alkyl of 1 to 5 carbon atoms and R.sub.3 is arylsulfonyl which possess ant…

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.