Patent · US Expired

Ibuprofen p-hydroxyphenylurea ester

US4049700A · kind A · utility

7Cited by
1References
1Claims
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Assignee

Inventor

Key dates

Filing dateJun 17, 1976
Grant dateSep 20, 1977
Priority date
Expiry dateJun 17, 1996

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P29/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Ibuprofen p-hydroxyphenylurea ester having the formula II: ##STR1## was prepared from the free acid, ibuprofen [.+-.2-(p-isobutylphenyl)propionic acid](I). The ester II above has the anti-inflammatory activity of the free acid, but in contradistinction to it, it has a pleasant taste, suitable for oral administration such as uncoated tablets, suspensions or syrups, for the treatment of inflammatory conditions, particularly arthritis.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.