Patent · US Expired

Process for the preparation of 6-alkoxy-substituted penicillins

US4051126A · kind A · utility

4Cited by
3References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 13, 1976
Grant dateSep 27, 1977
Priority date
Expiry dateJul 13, 1996

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D499/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

An improved process of preparing a 6-alkoxy-substituted penicillin or penicillin sulfoxide is disclosed. This process comprises adding a halogenating agent to penicillin or penicillin sulfoxide while cooling, and then adding an alkali metal alcoholate to the hydrogenation product in the presence of an alcohol corresponding to the alcoholate.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.