Patent · US Expired

1-(Arylamino)-and 1-(arylimino)-pyrroles

US4051147A · kind A · utility

6Cited by
1References
12Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJun 9, 1975
Grant dateSep 27, 1977
Priority date
Expiry dateJun 9, 1995

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D207/50
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

1-(Arylamino)pyrroles and 1-(arylimino)pyrroles, useful as antibacterial agents, are prepared by reaction of an arylhydrazine or arylhydrazone with a 2,5-di-lower-alkoxytetrahydrofuran or with an alkanedione; by reaction of a 1-arylaminopyrrole with an oxalyl dihalide followed by oxidative hydrolysis of the product; by condensation of a 1-aminopyrrole with a quinone; or by oxidation or reduction of a respective 1-(arylamino)pyrrole or 1-(arylimino)pyrrole.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.