Patent · US Expired

1-[2-(.beta.Naphthyloxy)ethyl]-3-methylpyrazolone-(5) and antithrombotic and antithrombolytic compositions and methods utilizing them

US4053621A · kind A · utility

5Cited by
26References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 2, 1975
Grant dateOct 11, 1977
Priority date
Expiry dateJun 2, 1995

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D231/20
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

1-[2-(.beta.-Naphthyloxy)ethyl]-3-methylpyrazolone-(5) and its salts are useful in the treatment and prophylaxis of thrombotic conditions. The compound is prepared through the reaction of 2-(.beta.-naphthyloxy)ethylhydrazine with either an acetoacetate or an ester of tetrolic acid, or through the condensation of 3-methylpyrazolinone-(5) with a derivative of 2-(.beta.-naphthyloxy)ethane, optionally with subsequent salt formation.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.