Patent · US Expired

Alpha-aryl-2-pyridineethanol 1-oxides and alpha-pyridinyl-2-pyridineethanol 1-oxides

US4056532A · kind A · utility

1Cited by
0References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 24, 1976
Grant dateNov 1, 1977
Priority date
Expiry dateJun 24, 1996

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D213/89
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Alpha-aryl-2-pyridineethanol 1-oxides and alpha-pyridinyl-2-pyridineethanol 1-oxides having the formula I or II: ##STR1## wherein R.sub.1 is hydrogen, halogen, hydroxy, lower alkyl, lower alkoxy, benzyloxy, lower alkanoyloxy, ortho-amino or ortho-lower alkylamino; R.sub.2 and R.sub.3 are each hydrogen, halogen, hydroxy, lower alkyl, lower alkoxy, benzyloxy or lower alkanoyloxy; the pharmaceutically acceptable acid addition salts thereof and a process for the preparation thereof are described. The compounds of this invention are useful in the prevention of allergic and asthmatic reactions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.